PDB entry 3gwt
View 3gwt on RCSB PDB site
Description: Catalytic domain of human phosphodiesterase 4B2B in complex with a quinoline inhibitor
Class: hydrolase
Keywords: PDE, PHOSPHODIESTERASE, cAMP, Hydrolase
Deposited on
2009-04-01, released
2010-04-07
The last revision prior to the SCOPe 2.06 freeze date was dated
2010-04-07, with a file datestamp of
2010-04-02.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: 0.207
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-specific 3',5'-cyclic phosphodiesterase 4B
Species: Homo sapiens [TaxId:9606]
Gene: PDE4B, DPDE4
Database cross-references and differences (RAF-indexed):
- Uniprot Q07343 (1-End)
- engineered (331)
- engineered (336)
Domains in SCOPe 2.06: d3gwta_ - Heterogens: 066, ZN, MG, ARS, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3gwtA (A:)
msisrfgvntenedhlakeledlnkwglnifnvagyshnrpltcimyaifqerdllktfr
issdtfitymmtledhyhsdvayhnslhaadvaqsthvllstpaldavftdleilaaifa
aaihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqeehcdifmnltkkq
rqtlrkmvidmvlatdmskhmslladlktmvetkkvtssgvllldnytdriqvlrnmvhc
adlsnptkslelyrqwtdrimeeffqqgdkerergmeispmcdkhtasveksqvgfidyi
vhplwetwadlvqpdaqdildtlednrnwyqamipqapappldeqnrdcqglm
Sequence, based on observed residues (ATOM records): (download)
>3gwtA (A:)
sisrfgvntenedhlakeledlnkwglnifnvagyshnrpltcimyaifqerdllktfri
ssdtfitymmtledhyhsdvayhnslhaadvaqsthvllstpaldavftdleilaaifaa
aihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqeehcdifmnltkkqr
qtlrkmvidmvlatdmskhmslladlktmvetkkvtssgvllldnytdriqvlrnmvhca
dlsnptkslelyrqwtdrimeeffqqgdkerergmeispmcdkhtasveksqvgfidyiv
hplwetwadlvqpdaqdildtlednrnwyqamipqa