PDB entry 3g9l
View 3g9l on RCSB PDB site
Description: JNK3 bound to (Z)-1-((6-fluoro-4H-benzo[d][1,3]dioxin-8-yl)methyl)-3-(hydroxyimino)-4-styrylindolin-2-one
Class: transferase
Keywords: kinase, inhibitor, phosphorylation, ATP-binding, Epilepsy, Nucleotide-binding, Phosphoprotein, Serine/threonine-protein kinase, Transferase
Deposited on
2009-02-13, released
2009-04-28
The last revision prior to the SCOPe 2.01 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.222
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'X':
Compound: Mitogen-activated protein kinase 10
Species: Homo sapiens [TaxId:9606]
Gene: JNK3, JNK3A, MAPK10, PRKM10
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d3g9lx_ - Heterogens: J67, HOH
PDB Chain Sequences:
- Chain 'X':
Sequence, based on SEQRES records: (download)
>3g9lX (X:)
mgskskvdnqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsr
pfqnqthakrayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqvi
qmeldhermsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartagts
fmmtpyvvtryyrapevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvie
qlgtpcpefmkklqptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardlls
kmlvidpakrisvddalqhpyinvwydpaeveapppqiydkqlderehtieewkeliyke
vmnse
Sequence, based on observed residues (ATOM records): (download)
>3g9lX (X:)
nqfysvevgdstftvlkryqnlkpigivcaaydavldrnvaikklsrpfqnqthakrayr
elvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviqmeldhermsyll
yqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglsfmmtvtryyrapevilgmg
ykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieqlgtpcpefmkklqptvrnyve
nrpkyagltfpklfpdslfpadsehnklkasqardllskmlvidpakrisvddalqhpyi
nvwydpaeveapppqiderehtieewkeliykevmn