PDB entry 3g9l

View 3g9l on RCSB PDB site
Description: JNK3 bound to (Z)-1-((6-fluoro-4H-benzo[d][1,3]dioxin-8-yl)methyl)-3-(hydroxyimino)-4-styrylindolin-2-one
Class: transferase
Keywords: kinase, inhibitor, phosphorylation, ATP-binding, Epilepsy, Nucleotide-binding, Phosphoprotein, Serine/threonine-protein kinase, Transferase
Deposited on 2009-02-13, released 2009-04-28
The last revision prior to the SCOPe 2.01 freeze date was dated 2011-07-13, with a file datestamp of 2011-05-08.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.222
AEROSPACI score: 0.35 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'X':
    Compound: Mitogen-activated protein kinase 10
    Species: Homo sapiens [TaxId:9606]
    Gene: JNK3, JNK3A, MAPK10, PRKM10
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.01: d3g9lx_
  • Heterogens: J67, HOH

PDB Chain Sequences:

  • Chain 'X':
    Sequence, based on SEQRES records: (download)
    >3g9lX (X:)
    mgskskvdnqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsr
    pfqnqthakrayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqvi
    qmeldhermsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartagts
    fmmtpyvvtryyrapevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvie
    qlgtpcpefmkklqptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardlls
    kmlvidpakrisvddalqhpyinvwydpaeveapppqiydkqlderehtieewkeliyke
    vmnse
    

    Sequence, based on observed residues (ATOM records): (download)
    >3g9lX (X:)
    nqfysvevgdstftvlkryqnlkpigivcaaydavldrnvaikklsrpfqnqthakrayr
    elvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviqmeldhermsyll
    yqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglsfmmtvtryyrapevilgmg
    ykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieqlgtpcpefmkklqptvrnyve
    nrpkyagltfpklfpdslfpadsehnklkasqardllskmlvidpakrisvddalqhpyi
    nvwydpaeveapppqiderehtieewkeliykevmn