PDB entry 3f9n
View 3f9n on RCSB PDB site
Description: Crystal structure of chk1 kinase in complex with inhibitor 38
Class: transferase
Keywords: chek1, chk1, kinase, cell cycle checkpoint, ATP-binding, Cytoplasm, DNA damage, DNA repair, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase, Ubl conjugation
Deposited on
2008-11-14, released
2009-01-20
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-04-28, with a file datestamp of
2009-04-24.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.184
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3f9na_ - Heterogens: 38M, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3f9nA (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkgakrprvtsggvsespsgfskhiqsnldfs
pvnsasrtpgsgwskehhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3f9nA (A:)
edwdlvqtlggevqlavnrvteeavavkivdmknikkeicinkmlnhenvvkfyghrreg
niqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrdikpenll
lderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvdvwscgiv
ltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenpsaritip
dikkdrwynkplk