PDB entry 3efk
View 3efk on RCSB PDB site
Description: Structure of c-Met with pyrimidone inhibitor 50
Class: Transferase
Keywords: c-Met, Kinase inhibitor pyrimidone, Alternative splicing, ATP-binding, Chromosomal rearrangement, Disease mutation, Glycoprotein, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Polymorphism, Proto-oncogene, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2008-09-09, released
2008-10-07
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.257
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d3efka_ - Chain 'B':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d3efkb_ - Heterogens: MT4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3efkA (A:)
mqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkih
cavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlr
nfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfgla
rdmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypd
vntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig
ehyvhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3efkA (A:)
dlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihcavksln
ritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfirnet
hnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfpvkwmalesl
qtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyev
mlkcwhpkaemrpsfselvsrisaifstfigehyvh
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3efkB (B:)
mqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkih
cavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlr
nfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfgla
rdmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypd
vntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig
ehyvhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3efkB (B:)
dlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihcavksld
igevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfirnethnpt
vkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfpvkwmaleslqtqk
fttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyevmlkc
whpkaemrpsfselvsrisaifstfigehyvh