PDB entry 3dpk
View 3dpk on RCSB PDB site
Description: cFMS tyrosine kinase in complex with a pyridopyrimidinone inhibitor
Class: transferase
Keywords: RECEPTOR TYROSINE KINASE, KINASE-INHIBITOR COMPLEX, ATP-binding, Glycoprotein, Immunoglobulin domain, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Polymorphism, Proto-oncogene, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase, Alternative splicing, Chromosomal rearrangement, Craniosynostosis, Disease mutation, Dwarfism, Heparin-binding, Kallmann syndrome
Deposited on
2008-07-08, released
2009-02-17
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-06-30, with a file datestamp of
2009-06-26.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.192
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Macrophage colony-stimulating factor 1 receptor
Species: Homo sapiens [TaxId:9606]
Gene: CSF1R, FMS, FGFR1, FGFBR, FLG, FLT2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3dpka_ - Heterogens: SO4, 8C5, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3dpkA (A:)
gvdykykqkpkyqvrwkiiesyegnsytfidptqlpynekwefprnnlqfgktlgagafg
kvveatafglgkedavlkvavkmlkstahadekealmselkimshlgqhenivnllgact
hggpvlviteyccygdllnflrrkrppgleysynpshnpeeqlssrdllhfssqvaqgma
flaskncihrdvaarnvlltnghvakigdfglardimndsnyivkgnarlpvkwmapesi
fdcvytvqsdvwsygillweifslglnpypgilvnskfyklvkdgyqmaqpafapkniys
imqacwalepthrptfqqicsflqeqaqedrrerd
Sequence, based on observed residues (ATOM records): (download)
>3dpkA (A:)
vrwkiiessytfidpynekwefprnnlqfgktlgagafgkvveatafglgavlkvavkml
kstahadekealmselkimshlgqhenivnllgacthggpvlviteyccygdllnflrrq
lssrdllhfssqvaqgmaflaskncihrdvaarnvlltnghvakigdfglardimndsny
ivrlpvkwmapesifdcvytvqsdvwsygillweifslglnpypgilvnskfyklvkdgy
qmaqpafapkniysimqacwalepthrptfqqicsflqe