PDB entry 3bgq
View 3bgq on RCSB PDB site
Description: Human Pim-1 kinase in complex with an triazolo pyridazine inhibitor VX2
Class: Transferase
Keywords: kinase inhibitor phosphorylation, Alternative initiation, ATP-binding, Cytoplasm, Manganese, Membrane, Metal-binding, Nucleotide-binding, Nucleus, Phosphoprotein, Proto-oncogene, Serine/threonine-protein kinase, Transferase
Deposited on
2007-11-27, released
2007-12-11
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.213
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene serine/threonine-protein kinase Pim-1
Species: Homo sapiens [TaxId:9606]
Gene: PIM1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d3bgqa1 - Heterogens: VX2, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3bgqA (A:)
mgsshhhhhhssglvprgshmllskinslahlraapcndlhatklapgkekeplesqyqv
gpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvllkkvssgf
sgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvleavrhchn
cgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppewiryhryhg
rsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwclalrpsdrpt
feeiqnhpwmqdvllpqetaeihlhslspgpsk
Sequence, based on observed residues (ATOM records): (download)
>3bgqA (A:)
plesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvl
lkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvl
eavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppew
iryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcla
lrpsdrptfeeiqnhpwmqdvllpqetaeihlh