PDB entry 3b65
View 3b65 on RCSB PDB site
Description: Crystal structure of the androgen receptor ligand binding domain in complex with SARM S-24
Class: transcription
Keywords: androgen receptor, sarm, Disease mutation, DNA-binding, Lipid-binding, Metal-binding, Nucleus, Polymorphism, Steroid-binding, Transcription, Transcription regulation, Triplet repeat expansion, Ubl conjugation, Zinc, Zinc-finger
Deposited on
2007-10-27, released
2008-09-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.242
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Androgen receptor
Species: Homo sapiens [TaxId:9606]
Gene: AR, DHTR, NR3C4
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3b65a_ - Heterogens: 3B6, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3b65A (A:)
piflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlhv
ddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksrmysqcvrmrhl
sqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrknpt
scsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsgk
vkpiyfhtq
Sequence, based on observed residues (ATOM records): (download)
>3b65A (A:)
piflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlhv
ddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksrmysqcvrmrhl
sqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrknpt
scsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsgk
vkpiyfh