PDB entry 3am4
View 3am4 on RCSB PDB site
Description: A372M mutant of Enoyl-ACP Reductase from Plasmodium falciparum (PfENR) in complex with triclosan variant T1
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: Triclosan, Triclosan variant, Enoyl-ACP reductase, mutant, oxidoreductase, P.falciparum, FabI, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2010-08-14, released
2011-03-16
The last revision prior to the SCOPe 2.08 freeze date was dated
2012-02-29, with a file datestamp of
2012-02-24.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.211
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Enoyl-ACP reductase
Species: Plasmodium falciparum [TaxId:5833]
Gene: FabI
Database cross-references and differences (RAF-indexed):
- Uniprot Q9BJJ9 (0-328)
- engineered mutation (276)
Domains in SCOPe 2.08: d3am4a_ - Chain 'B':
Compound: Enoyl-ACP reductase
Species: Plasmodium falciparum [TaxId:5833]
Gene: FabI
Database cross-references and differences (RAF-indexed):
- Uniprot Q9BJJ9 (0-328)
- engineered mutation (276)
Domains in SCOPe 2.08: d3am4b_ - Heterogens: NAD, FT1, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3am4A (A:)
nedicfiagigdtngygwgiakelskrnvkiifgiwppvynifmknykngkfdndmiidk
dkkmnildmlpfdasfdtandideetknnkrynmlqnytiedvanlihqkygkinmlvhs
lanakevqkdllntsrkgyldalskssyslislckyfvnimkpqssiisltyhasqkvvp
gygggmssakaalesdtrvlayhlgrnynirintisagplksraatainklnntyenntn
qnknrnrhdvhnimnnsgekeekkisasqnytfidymieysekyaplrqkllstdigsva
sfllsresraitgqtiyvdnglnimflpd
Sequence, based on observed residues (ATOM records): (download)
>3am4A (A:)
nedicfiagigdtngygwgiakelskrnvkiifgiwppvynifmknykngkfdndmiidk
dkkmnildmlpfdasfdtandideetknnkrynmlqnytiedvanlihqkygkinmlvhs
lanakevqkdllntsrkgyldalskssyslislckyfvnimkpqssiisltyhasqkvvp
gygggmssakaalesdtrvlayhlgrnynirintisagplksraataintfidymieyse
kyaplrqkllstdigsvasfllsresraitgqtiyvdnglnimflpd
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3am4B (B:)
nedicfiagigdtngygwgiakelskrnvkiifgiwppvynifmknykngkfdndmiidk
dkkmnildmlpfdasfdtandideetknnkrynmlqnytiedvanlihqkygkinmlvhs
lanakevqkdllntsrkgyldalskssyslislckyfvnimkpqssiisltyhasqkvvp
gygggmssakaalesdtrvlayhlgrnynirintisagplksraatainklnntyenntn
qnknrnrhdvhnimnnsgekeekkisasqnytfidymieysekyaplrqkllstdigsva
sfllsresraitgqtiyvdnglnimflpd
Sequence, based on observed residues (ATOM records): (download)
>3am4B (B:)
nedicfiagigdtngygwgiakelskrnvkiifgiwppvynifmknykngkfdndmiidk
dkkmnildmlpfdasfdtandideetknnkrynmlqnytiedvanlihqkygkinmlvhs
lanakevqkdllntsrkgyldalskssyslislckyfvnimkpqssiisltyhasqkvvp
gygggmssakaalesdtrvlayhlgrnynirintisagplksraataintfidymieyse
kyaplrqkllstdigsvasfllsresraitgqtiyvdnglnimflpd