PDB entry 3a4p
View 3a4p on RCSB PDB site
Description: human c-MET kinase domain complexed with 6-benzyloxyquinoline inhibitor
Class: Transferase
Keywords: C-MET, TYROSINE-PROTEIN KINASE, HEPATOCYTE GROWTH FACTOR RECEPTOR, Transferase
Deposited on
2009-07-13, released
2010-02-16
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2.54 Å
R-factor: 0.183
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3a4pa_ - Heterogens: CL, IPA, DFQ, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3a4pA (A:)
gplhmgsntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldnd
gkkihcavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymk
hgdlrnfirnethnptvkdligfglqvakgmkflaskkfvhrdlaarncmldekftvkva
dfglardmydkefdsvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrga
ppypdvntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaif
stfigehyvhvnatyvnvk
Sequence, based on observed residues (ATOM records): (download)
>3a4pA (A:)
vqavqhvvigpsslivhfnevigrghfgcvyhgtlldkkihcavkslnritdigevsqfl
tegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfirnethnptvkdligfg
lqvakgmkflaskkfvhrdlaarncmldekftvkvadfglardmydkaklpvkwmalesl
qtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyev
mlkcwhpkaemrpsfselvsrisaifstfigehyvhvnatyvnvk