PDB entry 2zmi
View 2zmi on RCSB PDB site
Description: Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism
Class: transcription
Keywords: NUCLEAR RECEPTOR-ANTAGONIST COMPLEX, DNA-binding, Metal-binding, Nucleus, Phosphoprotein, Receptor, Transcription, Transcription regulation, Zinc, Zinc-finger, Activator
Deposited on
2008-04-19, released
2008-09-02
The last revision prior to the SCOP 1.75 freeze date was dated
2008-09-16, with a file datestamp of
2008-09-12.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: 0.212
AEROSPACI score: 0.66
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Vitamin D3 receptor
Species: Rattus norvegicus [TaxId:10116]
Gene: Vdr, Nr1i1
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.75: d2zmia1 - Chain 'C':
Compound: Mediator of RNA polymerase II transcription subunit 1
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: TT2, EDO, FMT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2zmiA (A:)
gshmgspnsplkdslrpklseeqqhiiailldahhktydptyadfrdfrppvrmdgstgs
vtldlsplsmlphladlvsysiqkvigfakmipgfrdltsddqivllkssaievimlrsn
qsftmddmswdcgsqdykydvtdvskaghtlelieplikfqvglkklnlheeehvllmai
civspdrpgvqdaklveaiqdrlsntlqtyircrhpppgshqlyakmiqkladlrslnee
hskqyrslsfqpensmkltplvlevfgneis
Sequence, based on observed residues (ATOM records): (download)
>2zmiA (A:)
rpklseeqqhiiailldahhktydptyadfrdfrppvrmsplsmlphladlvsysiqkvi
gfakmipgfrdltsddqivllkssaievimlrsnqsftmddmswdcgsqdykydvtdvsk
aghtlelieplikfqvglkklnlheeehvllmaicivspdrpgvqdaklveaiqdrlsnt
lqtyircrhpppgshqlyakmiqkladlrslneehskqyrslsfqpensmkltplvlevf
gn
- Chain 'C':
No sequence available.