PDB entry 2zmd
View 2zmd on RCSB PDB site
Description: Crystal structure of human Mps1 catalytic domain T686A mutant in complex with SP600125 inhibitor
Class: transferase
Keywords: kinase, Mps1, SP600125, T686A, ATP-binding, Nucleotide-binding, Phosphoprotein, Serine/threonine-protein kinase, Transferase, Tyrosine-protein kinase
Deposited on
2008-04-16, released
2008-05-13
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2.88 Å
R-factor: 0.223
AEROSPACI score: 0.26
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dual specificity protein kinase TTK
Species: Homo sapiens [TaxId:9606]
Gene: TTK, MPS1L1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d2zmda_ - Heterogens: 537, 7PE, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2zmdA (A:)
hhhhhhssglvprgsgmketaaakferqhmdspdlgtddddkasssanecisvkgriysi
lkqigsggsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiaylnklqqhsdkiir
lydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmleavhtihqhgivhsd
lkpanflivdgmlklidfgianqmqpdttsvvkdsqvgavnymppeaikdmsssrengks
kskispksdvwslgcilyymtygktpfqqiinqisklhaiidpnheiefpdipekdlqdv
lkcclkrdpkqrisipellahpyvqiqthpvnqmakgtteemkyvlgqlvglnspnsilk
aaktlyehysggeshnssssktfekkrgkk
Sequence, based on observed residues (ATOM records): (download)
>2zmdA (A:)
ecisvkgriysilkqigsggsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiayl
nklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmleav
htihqhgivhsdlkpanflivdgmlklidfgianqmdsqvgavnymppeaikdmispksd
vwslgcilyymtygktpfqqiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdp
kqrisipellahpyvqiqt