PDB entry 2zlc
View 2zlc on RCSB PDB site
Description: 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure
Class: hormone
Keywords: Protein-ligand complex, DNA-binding, Metal-binding, Nucleus, Phosphoprotein, Receptor, Transcription, Transcription regulation, Zinc, Zinc-finger, HORMONE
Deposited on
2008-04-04, released
2008-06-24
The last revision prior to the SCOP 1.75 freeze date was dated
2008-08-12, with a file datestamp of
2008-08-08.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.225
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Vitamin D3 receptor
Species: Rattus norvegicus [TaxId:10116]
Gene: Vdr, Nr1i1
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.75: d2zlca1 - Chain 'C':
Compound: Coactivator peptide DRIP
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: VDX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2zlcA (A:)
gshmgspnsplkdslrpklseeqqhiiailldahhktydptyadfrdfrppvrmdgstgs
vtldlsplsmlphladlvsysiqkvigfakmipgfrdltsddqivllkssaievimlrsn
qsftmddmswdcgsqdykydvtdvskaghtlelieplikfqvglkklnlheeehvllmai
civspdrpgvqdaklveaiqdrlsntlqtyircrhpppgshqlyakmiqkladlrslnee
hskqyrslsfqpensmkltplvlevfgneis
Sequence, based on observed residues (ATOM records): (download)
>2zlcA (A:)
klseeqqhiiailldahhktydptyadfrdfrppvrmsplsmlphladlvsysiqkvigf
akmipgfrdltsddqivllkssaievimlrsnqsftmddmswdcgsqdykydvtdvskag
htlelieplikfqvglkklnlheeehvllmaicivspdrpgvqdaklveaiqdrlsntlq
tyircrhpppgshqlyakmiqkladlrslneehskqyrslsfqpensmkltplvlevfgn
- Chain 'C':
No sequence available.