PDB entry 2wgj
View 2wgj on RCSB PDB site
Description: x-ray structure of pf-02341066 bound to the kinase domain of c-met
Class: transferase
Keywords: c-met, kinase, inhibitor, transferase, ATP-binding, nucleotide-binding, tyrosine-protein kinase
Deposited on
2009-04-20, released
2009-06-02
The last revision prior to the SCOPe 2.03 freeze date was dated
2011-09-28, with a file datestamp of
2011-09-23.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.21485
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d2wgja_ - Heterogens: VGH, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2wgjA (A:)
mvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihcav
kslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfi
rnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfglardm
ydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdvnt
fditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfigehh
hhhhhh
Sequence, based on observed residues (ATOM records): (download)
>2wgjA (A:)
hidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtllkkihcavkslnri
tdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfirnethn
ptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfglardmydkeyy
svhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdvntfditvy
llqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfi