PDB entry 2w8y
View 2w8y on RCSB PDB site
Description: ru486 bound to the progesterone receptor in a destabilized agonistic conformation
Class: receptor
Keywords: receptor, progesterone receptor, ru-486, mifepristone
Deposited on
2009-01-20, released
2009-04-28
The last revision prior to the SCOPe 2.05 freeze date was dated
2011-07-13, with a file datestamp of
2011-06-02.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.187
AEROSPACI score: 0.54
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: progesterone receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- PDB 2W8Y
- Uniprot P06401 (Start-259)
Domains in SCOPe 2.05: d2w8ya_ - Chain 'B':
Compound: progesterone receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- PDB 2W8Y
- Uniprot P06401 (Start-259)
Domains in SCOPe 2.05: d2w8yb_ - Heterogens: 486, SO4, NDR, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2w8yA (A:)
gshmgqdiqlipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkws
kslpgfrnlhiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkess
fyslcltmwqipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyireli
kaiglrqkgvvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmsevi
aaqlpkilagmvkpllfhkk
Sequence, based on observed residues (ATOM records): (download)
>2w8yA (A:)
lipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkwskslpgfrnl
hiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkessfyslcltmw
qipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyirelikaiglrqkg
vvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmseviaaqlpkila
gmvkpllfhkk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2w8yB (B:)
gshmgqdiqlipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkws
kslpgfrnlhiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkess
fyslcltmwqipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyireli
kaiglrqkgvvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmsevi
aaqlpkilagmvkpllfhkk
Sequence, based on observed residues (ATOM records): (download)
>2w8yB (B:)
lipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkwskslpgfrnl
hiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkessfyslcltmw
qipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyirelikaiglrqkg
vvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmseviaaqlpkila
gmvkpllfhkk