PDB entry 2qyk
View 2qyk on RCSB PDB site
Description: Crystal structure of PDE4A10 in complex with inhibitor NPV
Class: hydrolase
Keywords: PDE4 inhibitor, subfamily inhibitor selectivity, Hydrolase
Deposited on
2007-08-15, released
2008-04-08
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.201
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Cyclic AMP-specific phosphodiesterase HSPDE4A10
Species: Homo sapiens [TaxId:9606]
Gene: PDE4A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2qyka1, d2qyka2 - Chain 'B':
Compound: Cyclic AMP-specific phosphodiesterase HSPDE4A10
Species: Homo sapiens [TaxId:9606]
Gene: PDE4A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2qykb1, d2qykb2 - Heterogens: NPV, ZN, MG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2qykA (A:)
hmniprfgvktdqeellaqelenlnkwglnifcvsdyaggrsltcimymifqerdllkkf
ripvdtmvtymltledhyhadvayhnslhaadvlqsthvllatpaldavftdleilaalf
aaaihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqedncdifqnlskr
qrqslrkmvidmvlatdmskhmtlladlktmvetkkvtssgvllldnysdriqvlrnmvh
cadlsnptkplelyrqwtdrimaeffqqgdrerergmeispmcdkhtasveksqvgfidy
ivhplwetwadlvhpdaqeildtlednrdwyysai
Sequence, based on observed residues (ATOM records): (download)
>2qykA (A:)
mniprfgvktdqeellaqelenlnkwglnifcvsdyaggrsltcimymifqerdllkkfr
ipvdtmvtymltledhyhadvayhnslhaadvlqsthvllatpaldavftdleilaalfa
aaihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqedncdifqnlskrq
rqslrkmvidmvlatdmskhmtlladlktmvetkkvtssgvllldnysdriqvlrnmvhc
adlsnptkplelyrqwtdrimaeffqqgdrerergmeispmcdkhtasveksqvgfidyi
vhplwetwadlvhpdaqeildtlednrdwyysai
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>2qykB (B:)
hmniprfgvktdqeellaqelenlnkwglnifcvsdyaggrsltcimymifqerdllkkf
ripvdtmvtymltledhyhadvayhnslhaadvlqsthvllatpaldavftdleilaalf
aaaihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqedncdifqnlskr
qrqslrkmvidmvlatdmskhmtlladlktmvetkkvtssgvllldnysdriqvlrnmvh
cadlsnptkplelyrqwtdrimaeffqqgdrerergmeispmcdkhtasveksqvgfidy
ivhplwetwadlvhpdaqeildtlednrdwyysai