PDB entry 2p15
View 2p15 on RCSB PDB site
Description: Crystal structure of the ER alpha ligand binding domain with the agonist ortho-trifluoromethylphenylvinyl estradiol
Class: hormone receptor
Keywords: nulear receptor, ligand binding domain, helix 12, HORMONE RECEPTOR
Deposited on
2007-03-02, released
2007-05-01
The last revision prior to the SCOPe 2.01 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 1.94 Å
R-factor: 0.161
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Gene: ESR1, ESR, NR3A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d2p15a_ - Chain 'B':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Gene: ESR1, ESR, NR3A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d2p15b_ - Chain 'C':
Compound: GRIP peptide
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'D':
Compound: GRIP peptide
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: EZT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2p15A (A:)
sikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvh
minwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgk
cvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhih
rvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpl
sdlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>2p15A (A:)
slalsltadqmvsalldaeppilyseyrpfseasmmglltnladrelvhminwakrvpgf
vdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmveifdm
llatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitdtli
hlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplsdlllemldah
rl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2p15B (B:)
sikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvh
minwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgk
cvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhih
rvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpl
sdlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>2p15B (B:)
lalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrvp
gfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmveif
dmllatssrfrmmnlqgeefvclksiillnsgvytftlksleekdhihrvldkitdtlih
lmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplsdlllemldahr
lh
- Chain 'C':
No sequence available.
- Chain 'D':
No sequence available.