PDB entry 2obj
View 2obj on RCSB PDB site
Description: Crystal structure of human PIM-1 Kinase in complex with inhibitor
Class: transferase
Keywords: PIM, PIM-1, PIM1, human PIM-1 Kinase, Serine/threonine kinase, kinase inhibitor complex, Pyridone, kinase inhibitor
Deposited on
2006-12-19, released
2007-02-06
The last revision prior to the SCOP 1.73 freeze date was dated
2007-03-06, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.205
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene serine/threonine-protein kinase Pim-1
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d2obja1 - Heterogens: VRV, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2objA (A:)
mgsshhhhhhssglvprgshmllskinslahlraapcndlhatklapgkekeplesqyqv
gpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvllkkvssgf
sgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvleavrhchn
cgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppewiryhryhg
rsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwclalrpsdrpt
feeiqnhpwmqdvllpqetaeihlhslspgpsk
Sequence, based on observed residues (ATOM records): (download)
>2objA (A:)
plesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvl
lkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvl
eavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppew
iryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcla
lrpsdrptfeeiqnhpwmqdvllpqetaeihlh