PDB entry 2jdr
View 2jdr on RCSB PDB site
Description: structure of pkb-beta (akt2) complexed with the inhibitor a-443654
Class: transferase
Keywords: wnt signaling pathway, serine/threonine-protein kinase, kinase, transferase, ATP-binding, phosphorylation, nucleotide-binding, alternative splicing
Deposited on
2007-01-12, released
2007-02-13
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.196
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: rac-beta serine/threonine-protein kinase
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- PDB 2JDR (Start-341)
- Uniprot P31751 (5-End)
Domains in SCOPe 2.08: d2jdra_ - Chain 'C':
Compound: Glycogen synthase kinase-3 beta
Species: HOMO SAPIENS, synthetic [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Heterogens: L20, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2jdrA (A:)
gamdpkvtmndfdylkllgkgtfgkvilvrekatgryyamkilrkeviiakdevahtvte
srvlqntrhpfltalkyafqthdrlcfvmeyanggelffhlsrervfteerarfygaeiv
saleylhsrdvvyrdiklenlmldkdghikitdfglckegisdgatmktfcgtpeylape
vledndygravdwwglgvvmyemmcgrlpfynqdherlfelilmeeirfprtlspeaksl
lagllkkdpkqrlgggpsdakevmehrfflsinwqdvvqkkllppfkpqvtsevdtryfd
deftaqsititppdrydslglleldqreeqemfedfdyiadw
Sequence, based on observed residues (ATOM records): (download)
>2jdrA (A:)
kvtmndfdylkllgkgtfgkvilvrekatgryyamkilrkeviiakdevahtvtesrvlq
ntrhpfltalkyafqthdrlcfvmeyanggelffhlsrervfteerarfygaeivsaley
lhsrdvvyrdiklenlmldkdghikitdfglckegisdgatmktfcgtpeylapevledn
dygravdwwglgvvmyemmcgrlpfynqdherlfelilmeeirfprtlspeaksllagll
kkdpkqrlgggpsdakevmehrfflsinwqdvvqkkllppfkpqvtsevdtryfddefta
qsitqemfedfdyiadw
- Chain 'C':
No sequence available.