PDB entry 2f81
View 2f81 on RCSB PDB site
Description: HIV-1 Protease mutant L90M complexed with inhibitor TMC114
Class: hydrolase
Keywords: HIV-1 protease-inhibitor complex, HYDROLASE
Deposited on
2005-12-01, released
2006-03-07
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-18, with a file datestamp of
2017-10-13.
Experiment type: XRAY
Resolution: 1.25 Å
R-factor: N/A
AEROSPACI score: 0.62
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Pol polyprotein
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot P04587
- engineered (6)
- engineered (32)
- engineered (62)
- engineered (66)
- engineered (89)
- engineered (94)
Domains in SCOPe 2.08: d2f81a_ - Chain 'B':
Compound: Pol polyprotein
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot P04587 (0-98)
- engineered (6)
- engineered (32)
- engineered (62)
- engineered (66)
- engineered (89)
- engineered (94)
Domains in SCOPe 2.08: d2f81b_ - Heterogens: NA, CL, 017, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>2f81A (A:)
pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpkmiggiggfikvrqyd
qiiieiaghkaigtvlvgptpvniigrnlmtqigatlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>2f81B (B:)
pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpkmiggiggfikvrqyd
qiiieiaghkaigtvlvgptpvniigrnlmtqigatlnf