PDB entry 2bzh
View 2bzh on RCSB PDB site
Description: crystal structure of the human pim1 in complex with a ruthenium organometallic ligand ru1
Class: transferase
Keywords: pim1, kinase, cancer, leukemia, nuclear protein, nucleotide-binding, transferase
Deposited on
2005-08-18, released
2005-12-08
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-31.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.159
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'B':
Compound: proto-oncogene serine threonine protein kinase pim1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P11309
- engineered mutation (249)
Domains in SCOPe 2.06: d2bzhb_ - Heterogens: HB1, EDO, CL, HOH
PDB Chain Sequences:
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2bzhB (B:)
mllskinslahlraapcndlhatklapgkekeplesqyqvgpllgsggfgsvysgirvsd
nlpvaikhvekdrisdwgelpngtrvpmevvllkkvssgfsgvirlldwferpdsfvlil
erpepvqdlfdfitergalqeelarsffwqvleavrhchncgvlhrdikdenilidlnrg
elklidfgsgallkdtvytdfdgtrvysppewiryhryhgrsaavwslgillydmvcgdi
pfehdeeiiggqvffrqrvssecqhlirwclalrpsdrptfeeiqnhpwmqdvllpqeta
eihlhslspgpsk
Sequence, based on observed residues (ATOM records): (download)
>2bzhB (B:)
eplesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevv
llkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqv
leavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppe
wiryhryhgrsaavwslgillydmvcgdipfehdeeiiggqvffrqrvssecqhlirwcl
alrpsdrptfeeiqnhpwmqdvllpqetaeihlhs