PDB entry 2bdj
View 2bdj on RCSB PDB site
Description: Src kinase in complex with inhibitor AP23464
Class: transferase
Keywords: Src kinase
Inhibitor
Deposited on
2005-10-20, released
2006-10-24
The last revision prior to the SCOP 1.73 freeze date was dated
2006-10-24, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.158
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: HOMO SAPIENS
Gene: SRC, SRC1
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d2bdja1 - Heterogens: HET, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2bdjA (A:)
lakdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaflqeaqvm
kklrheklvqlyavvseepiyivteymskgslldflkgetgkylrlpqlvdmaaqiasgm
ayvermnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpikwtapeaa
lygrftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppecpeslhdl
mcqcwrkepeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>2bdjA (A:)
kdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaflqeaqvmkk
lrheklvqlyavvseepiyivteymskgslldflkgetgkylrlpqlvdmaaqiasgmay
vermnyvhrdlraanilvgenlvckvadfglarliefpikwtapeaalygrftiksdvws
fgilltelttkgrvpypgmvnrevldqvergyrmpcppecpeslhdlmcqcwrkepeerp
tfeylqafledyft