PDB entry 2agt

View 2agt on RCSB PDB site
Description: Aldose Reductase Mutant Leu 300 Pro complexed with Fidarestat
Class: oxidoreductase
Keywords: OXIDOREDUCTASE, NADP, Fidarestat,
Deposited on 2005-07-27, released 2005-09-20
The last revision prior to the SCOPe 2.08 freeze date was dated 2009-02-24, with a file datestamp of 2009-03-01.
Experiment type: XRAY
Resolution: 1 Å
R-factor: 0.106
AEROSPACI score: 1.04 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: aldose reductase
    Species: Homo sapiens [TaxId:9606]
    Gene: AKR1B1, ALDR1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P15121 (3-318)
      • engineered (303)
    Domains in SCOPe 2.08: d2agta_
  • Heterogens: CL, NAP, FID, CIT, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >2agtA (A:)
    gshmasrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgv
    aiqeklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwptgfk
    pgkeffpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglk
    ykpavnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikai
    aakhnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwr
    vcaplsctshkdypfheef
    

    Sequence, based on observed residues (ATOM records): (download)
    >2agtA (A:)
    masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiq
    eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwptgfkpgk
    effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
    avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
    hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
    plsctshkdypfheef