PDB entry 1zoh
View 1zoh on RCSB PDB site
Description: Crystal structure of protein kinase CK2 in complex with TBB-derivatives inhibitors
Class: transferase
Keywords: Protein kinase CK2, tetrabromo-benzimidazole, TBB, inhibitors, pharmacophore
Deposited on
2005-05-13, released
2005-11-29
The last revision prior to the SCOP 1.75 freeze date was dated
2005-11-29, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 1.81 Å
R-factor: 0.165
AEROSPACI score: 0.59
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: protein kinase ck2, alpha subunit
Species: Zea mays
Gene: ACK2
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.75: d1zoha1 - Heterogens: NA, CL, K44, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1zohA (A:)
mskarvyadvnvlrpkeywdyealtvqwgeqddyevvrkvgrgkysevfeginvnnnekc
iikilkpvkkkkikreikilqnlcggpnivklldivrdqhsktpslifeyvnntdfkvly
ptltdydiryyiyellkaldychsqgimhrdvkphnvmidhelrklrlidwglaefyhpg
keynvrvasryfkgpellvdlqdydysldmwslgcmfagmifrkepffyghdnhdqlvki
akvlgtdglnvylnkyrieldpqlealvgrhsrkpwlkfmnadnqhlvspeaidfldkll
rydhqerltaleamthpyfqqvraaensrtra
Sequence, based on observed residues (ATOM records): (download)
>1zohA (A:)
mskarvyadvnvlrpkeywdyealtvqwgeqddyevvrkvgrgkysevfeginvnnnekc
iikilkpvkkkkikreikilqnlcggpnivklldivrdqhsktpslifeyvnntdfkvly
ptltdydiryyiyellkaldychsqgimhrdvkphnvmidhelrklrlidwglaefyhpg
keynvrvasryfkgpellvdlqdydysldmwslgcmfagmifrkepffyghdnhdqlvki
akvlgtdglnvylnkyrieldpqlealvgrhsrkpwlkfmnadnqhlvspeaidfldkll
rydhqerltaleamthpyfqqvraae