PDB entry 1yhv
View 1yhv on RCSB PDB site
Description: Crystal Structure of PAK1 kinase domain with two point mutations (K299R, T423E)
Class: signaling protein, transferase
Keywords: kinase; active conformation; activation loop; ATP binding site, SIGNALING PROTEIN, TRANSFERASE
Deposited on
2005-01-10, released
2005-05-24
The last revision prior to the SCOPe 2.03 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-19.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.22
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase PAK 1
Species: Homo sapiens [TaxId:9606]
Gene: PAK1
Database cross-references and differences (RAF-indexed):
- Uniprot Q13153 (0-End)
- engineered (50)
- engineered (174)
Domains in SCOPe 2.03: d1yhva_ - Heterogens: HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1yhvA (A:)
sdeeileklrsivsvgdpkkkytrfekigqgasgtvytamdvatgqevairqmnlqqqpk
keliineilvmrenknpnivnyldsylvgdelwvvmeylaggsltdvvtetcmdegqiaa
vcreclqaleflhsnqvihrdiksdnillgmdgsvkltdfgfcaqitpeqskrsemvgtp
ywmapevvtrkaygpkvdiwslgimaiemiegeppylnenplralyliatngtpelqnpe
klsaifrdflnrcldmdvekrgsakellqhqflkiakplssltpliaaakeatknnh
Sequence, based on observed residues (ATOM records): (download)
>1yhvA (A:)
sdeeileklrsivsvgdpkkkytrfekigqgasgtvytamdvatgqevairqmnlqqqpk
keliineilvmrenknpnivnyldsylvgdelwvvmeylaggsltdvvtetcmdegqiaa
vcreclqaleflhsnqvihrdiksdnillgmdgsvkltdfgfcaqitpeqskrsemvgtp
ywmapevvtrkaygpkvdiwslgimaiemiegeppylnenplralyliatngtpelqnpe
klsaifrdflnrcldmdvekrgsakellqhqflkiakplssltpliaaakeat