PDB entry 1xp0
View 1xp0 on RCSB PDB site
Description: Catalytic Domain Of Human Phosphodiesterase 5A In Complex With Vardenafil
Class: hydrolase
Keywords: Phosphodiesterase, PDE, PDE5A, Vardenafil, Levitra, HYDROLASE
Deposited on
2004-10-07, released
2004-12-14
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 1.79 Å
R-factor: 0.194
AEROSPACI score: 0.53
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cGMP-specific 3',5'-cyclic phosphodiesterase
Species: Homo sapiens [TaxId:9606]
Gene: PDE5A, PDE5
Database cross-references and differences (RAF-indexed):
- Uniprot O76074 (21-End)
- engineered (145)
- engineered (148)
- engineered (150)
- engineered (134-135)
- engineered (154-158)
- engineered (161-163)
- engineered (165-166)
- engineered (168-169)
Domains in SCOPe 2.06: d1xp0a_ - Heterogens: ZN, MG, VDN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1xp0A (A:)
mgsshhhhhhssglvprgshmeeetrelqslaaavvpsaqtlkitdfsfsdfelsdleta
lctirmftdlnlvqnfqmkhevlcrwilsvkknyrknvayhnwrhafntaqcmfaalkag
kiqnkltdleilalliaalshdldhpgvsnqflintnselalmyndesvlehhhfdqclm
ilnspgnqilsglsieeykttlkiikqailatdlalyikrrgeffelirknqfnledphq
kelflamlmtacdlsaitkpwpiqqriaelvateffdqgdrerkelnieptdlmnrekkn
kipsmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalaeqqekmlingesgq
akrn
Sequence, based on observed residues (ATOM records): (download)
>1xp0A (A:)
eeetrelqslaaavvpsaqtlkitdfsfsdfelsdletalctirmftdlnlvqnfqmkhe
vlcrwilsvkknyrknvayhnwrhafntaqcmfaalkagkiqnkltdleilalliaalsh
dldhpgvsnqflintnselalmyndesvlehhhfdqclmilnspgnqilsglsieeyktt
lkiikqailatdlalyikrrgeffelirknqfnledphqkelflamlmtacdlsaitkpw
piqqriaelvateffdqgdrerkelnieptdlmnrekknkipsmqvgfidaiclqlyeal
thvsedcfplldgcrknrqkwqalae