PDB entry 1vjy
View 1vjy on RCSB PDB site
Description: Crystal Structure of a Naphthyridine Inhibitor of Human TGF-beta Type I Receptor
Class: transferase
Keywords: transferase, protein kinase, Inhibitor Complex
Deposited on
2004-04-07, released
2004-08-31
The last revision prior to the SCOPe 2.03 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.223
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: tgf-beta receptor type I
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d1vjya_ - Heterogens: 460, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1vjyA (A:)
iartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhenil
gfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhmei
vgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkryma
pevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsvee
mrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqqeg
ikm
Sequence, based on observed residues (ATOM records): (download)
>1vjyA (A:)
iartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhenil
gfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhmei
vgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidirvgtkrymapevl
ddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsveemrkv
vceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqqegikm