PDB entry 1uom
View 1uom on RCSB PDB site
Description: the structure of estrogen receptor in complex with a selective and potent tetrahydroisochiolin ligand.
Class: nuclear protein
Keywords: selective estrogen receptor modulators, serm, receptor, transcription regulation, DNA-binding, nuclear protein, zinc-finger, steroid-binding, phosphorylation, polymorphism 3d-structure, alternative splicing
Deposited on
2003-04-11, released
2003-07-03
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.28 Å
R-factor: 0.235
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- PDB 1UOM
- engineered mutation (81)
- engineered mutation (117)
- Uniprot P03372
Domains in SCOPe 2.02: d1uoma_ - Heterogens: PTI, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1uomA (A:)
mskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhmin
wakrvpgfvdltlhdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksve
gmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvl
dkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmksknvvplydl
llemldahrlhapt
Sequence, based on observed residues (ATOM records): (download)
>1uomA (A:)
alsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrvpg
fvdltlhdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksvegmveifd
mllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitdtl
ihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlplydlllemldah