PDB entry 1o3p
View 1o3p on RCSB PDB site
Description: Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-Directed Serine Protease Inhibitors
Class: BLOOD CLOTTING, hydrolase
Keywords: serine protease, short hydrogen bond, inhibition mechanism, shift of pKa, trypsin, thrombin, urokinase, factor Xa, BLOOD CLOTTING, hydrolase
Deposited on
2003-03-06, released
2003-09-02
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-04, with a file datestamp of
2017-09-29.
Experiment type: XRAY
Resolution: 1.81 Å
R-factor: N/A
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: urokinase-type plasminogen activator
Species: Homo sapiens [TaxId:9606]
Gene: PLAU
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1o3p.1 - Chain 'B':
Compound: urokinase-type plasminogen activator
Species: Homo sapiens [TaxId:9606]
Gene: PLAU
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1o3p.1 - Heterogens: CIT, 655, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1o3pA (A:)
kpssppeelkfqcgqktlrprfk
Sequence, based on observed residues (ATOM records): (download)
>1o3pA (A:)
lkfqcgqk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>1o3pB (B:)
iiggefttienqpwfaaiyrrhrggsvtyvcggslmspcwvisathcfidypkkedyivy
lgrsrlnsntqgemkfevenlilhkdysadtlahhndiallkirskegrcaqpsrtiqti
clpsmyndpqfgtsceitgfgkeastdylypeqlkmtvvklishrecqqphyygsevttk
mlcaadpqwktdscqgdsggplvcslqgrmtltgivswgrgcalkdkpgvytrvshflpw
irshtkeenglal
Sequence, based on observed residues (ATOM records): (download)
>1o3pB (B:)
iiggefttienqpwfaaiyrrhrggsvtyvcggslmspcwvisathcfidypkkedyivy
lgrsrlnsntqgemkfevenlilhkdysadtlahhndiallkirskegrcaqpsrtiqti
clpsmyndpqfgtsceitgfgkeastdylypeqlkmtvvklishrecqqphyygsevttk
mlcaadpqwktdscqgdsggplvcslqgrmtltgivswgrgcalkdkpgvytrvshflpw
irshtk