PDB entry 1nwl
View 1nwl on RCSB PDB site
Description: Crystal structure of the PTP1B complexed with SP7343-SP7964, a pTyr mimetic
Class: hydrolase
Keywords: protein-small molecule inhibitor complex, HYDROLASE
Deposited on
2003-02-06, released
2003-04-01
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.21
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: protein-tyrosine phosphatase, non-receptor type 1
Species: Homo sapiens [TaxId:9606]
Gene: PTPN1
Database cross-references and differences (RAF-indexed):
- Uniprot P18031 (0-End)
- engineered (31)
- engineered (46)
- engineered (91)
Domains in SCOPe 2.02: d1nwla_ - Heterogens: MG, 964, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1nwlA (A:)
memekefeqidksgswaaiyqdirheasdfpsrvaklpknknrnrycdvspfdhsriklh
qedndyinaslikmeeaqrsyiltqgplpntvghfwemvweqksrgvvmlnrvmekgslk
caqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfhyttwp
dfgvpespasflnflfkvresgslspehgpvvvhcsagigrsgtfcladtclllmdkrkd
pssvdikkvllemrkfrmgliqtadqlrfsylaviegakfimgdssvqdqwkelshed
Sequence, based on observed residues (ATOM records): (download)
>1nwlA (A:)
memekefeqidksgswaaiyqdirheasdfpsrvaklpknknrnrycdvspfdhsriklh
qedndyinaslikmeeaqrsyiltqgplpntvghfwemvweqksrgvvmlnrvmekgslk
caqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfhyttwp
dfgvpespasflnflfkvresgslspehgpvvvhcsagigrsgtfcladtclllmdkrkd
pssvdikkvllemrkfrmgliqtadqlrfsylaviegakfimg