PDB entry 1m17
View 1m17 on RCSB PDB site
Description: Epidermal Growth Factor Receptor tyrosine kinase domain with 4-anilinoquinazoline inhibitor erlotinib
Class: transferase
Keywords: TRANSFERASE, tyrosine kinase domain
Deposited on
2002-06-17, released
2002-09-04
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.6 Å
R-factor: 0.251
AEROSPACI score: 0.25
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1m17a_ - Heterogens: AQ4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1m17A (A:)
gshmasgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelre
atspkankeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdni
gsqyllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekey
haeggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilek
gerlpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhl
psptdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>1m17A (A:)
geapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatspka
nkeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyll
nwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhaeggk
vpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpq
ppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlmdeedm
ddvvdadeylip