PDB entry 1l2i
View 1l2i on RCSB PDB site
Description: Human Estrogen Receptor alpha Ligand-binding Domain in Complex with (R,R)-5,11-cis-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol and a Glucocorticoid Receptor Interacting Protein 1 NR box II Peptide
Class: transcription receptor/coactivator
Keywords: nuclear receptor, transcription factor, estrogen, agonist, coactivator, TRANSCRIPTION RECEPTOR/COACTIVATOR COMPLEX
Deposited on
2002-02-21, released
2002-05-01
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.203
AEROSPACI score: 0.48
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d1l2ia_ - Chain 'B':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d1l2ib_ - Chain 'C':
Compound: glucocorticoid receptor-interacting protein 1
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'D':
Compound: glucocorticoid receptor-interacting protein 1
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: CL, ETC, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1l2iA (A:)
mdpmikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladre
lvhminwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrn
qgkcvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekd
hihrvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknv
vplydlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>1l2iA (A:)
slalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrv
pgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmvei
fdmllatssrfrmmnlqgeefvclksiillnsgvyleekdhihrvldkitdtlihlmaka
gltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplydlllemldah
- Chain 'B':
Sequence, based on SEQRES records: (download)
>1l2iB (B:)
mdpmikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladre
lvhminwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrn
qgkcvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekd
hihrvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknv
vplydlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>1l2iB (B:)
slalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrv
pgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmvei
fdmllatssrfrmmnlqgeefvclksiillnsgvytkdhihrvldkitdtlihlmakagl
tlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplydlllemldah
- Chain 'C':
No sequence available.
- Chain 'D':
No sequence available.