Lineage for d6vvpc_ (6vvp C:)

  1. Root: SCOPe 2.08
  2. 2685877Class a: All alpha proteins [46456] (290 folds)
  3. 2728284Fold a.123: Nuclear receptor ligand-binding domain [48507] (1 superfamily)
    multihelical; 3 layers or orthogonally packed helices
  4. 2728285Superfamily a.123.1: Nuclear receptor ligand-binding domain [48508] (2 families) (S)
  5. 2728286Family a.123.1.1: Nuclear receptor ligand-binding domain [48509] (34 proteins)
  6. 2728396Protein Estrogen receptor alpha [48519] (1 species)
  7. 2728397Species Human (Homo sapiens) [TaxId:9606] [48520] (107 PDB entries)
    Uniprot P03372 307-551
  8. 2728623Domain d6vvpc_: 6vvp C: [383264]
    automated match to d3q95b_
    complexed with r3v; mutant

Details for d6vvpc_

PDB Entry: 6vvp (more details), 2.6 Å

PDB Description: estrogen receptor alpha ligand binding domain y537s mutant in complex with a methylated lasofoxifene derivative that possesses selective estrogen receptor degrader activities
PDB Compounds: (C:) Estrogen receptor

SCOPe Domain Sequences for d6vvpc_:

Sequence, based on SEQRES records: (download)

>d6vvpc_ a.123.1.1 (C:) Estrogen receptor alpha {Human (Homo sapiens) [TaxId: 9606]}
lalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrvp
gfvdltlhdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksvegmveif
dmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitdt
lihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmksknvvplsdlllem

Sequence, based on observed residues (ATOM records): (download)

>d6vvpc_ a.123.1.1 (C:) Estrogen receptor alpha {Human (Homo sapiens) [TaxId: 9606]}
lalsltadqmvsalldaeppilyseydsmmglltnladrelvhminwakrvpgfvdltlh
dqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgkmveifdmllatssrfrm
mnlqgeefvclksiillnsgvyeekdhihrvldkitdtlihlmakagltlqqqhqrlaql
llilshirhmsnkgmehlysmsdlllem

SCOPe Domain Coordinates for d6vvpc_:

Click to download the PDB-style file with coordinates for d6vvpc_.
(The format of our PDB-style files is described here.)

Timeline for d6vvpc_: