Lineage for d3flia_ (3fli A:)

  1. Root: SCOPe 2.08
  2. 2685877Class a: All alpha proteins [46456] (290 folds)
  3. 2728284Fold a.123: Nuclear receptor ligand-binding domain [48507] (1 superfamily)
    multihelical; 3 layers or orthogonally packed helices
  4. 2728285Superfamily a.123.1: Nuclear receptor ligand-binding domain [48508] (2 families) (S)
  5. 2728286Family a.123.1.1: Nuclear receptor ligand-binding domain [48509] (34 proteins)
  6. 2728375Protein Bile acid receptor FXR [101433] (2 species)
  7. 2728376Species Human (Homo sapiens) [TaxId:9606] [101434] (8 PDB entries)
  8. 2728378Domain d3flia_: 3fli A: [175890]
    automated match to d1osha_
    complexed with 33y

Details for d3flia_

PDB Entry: 3fli (more details), 2 Å

PDB Description: Discovery of XL335, a Highly Potent, Selective and Orally-Active Agonist of the Farnesoid X Receptor (FXR)
PDB Compounds: (A:) Bile acid receptor

SCOPe Domain Sequences for d3flia_:

Sequence, based on SEQRES records: (download)

>d3flia_ a.123.1.1 (A:) Bile acid receptor FXR {Human (Homo sapiens) [TaxId: 9606]}
eltpdqqtllhfimdsynkqrmpqeitnkilkeefsaeenfliltematnhvqvlveftk
klpgfqtldhedqiallkgsaveamflrsaeifnkklpsghsdlleerirnsgisdeyit
pmfsfyksigelkmtqeeyalltaivilspdrqyikdreaveklqeplldvlqklckihq
penpqhfacllgrltelrtfnhhhaemlmswrvndhkftpllceiwdv

Sequence, based on observed residues (ATOM records): (download)

>d3flia_ a.123.1.1 (A:) Bile acid receptor FXR {Human (Homo sapiens) [TaxId: 9606]}
eltpdqqtllhfimdsynkqrmpqeitnkilkeefsaeenfliltematnhvqvlveftk
klpgfqtldhedqiallkgsaveamflrsaeifnkklpsghsdlleerirnsgisdeyit
pmfsfyksigelkmtqeeyalltaivilspdrqyikdreaveklqeplldvlqklckihq
penpqhfacllgrltelrtfnhhhaemlmsftpllceiwdv

SCOPe Domain Coordinates for d3flia_:

Click to download the PDB-style file with coordinates for d3flia_.
(The format of our PDB-style files is described here.)

Timeline for d3flia_: