PDB entry 7kpy
View 7kpy on RCSB PDB site
Description: Crystal structure of CBP bromodomain liganded with UMB298 (compound 23)
Class: transcription
Keywords: epigenetics, inhibitor, drug development, multi domain proteins, TRANSCRIPTION
Deposited on
2020-11-12, released
2021-05-19
The last revision prior to the SCOPe 2.08 freeze date was dated
2021-05-26, with a file datestamp of
2021-05-21.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: N/A
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: histone acetyltransferase
Species: Homo sapiens [TaxId:9606]
Gene: Crebbp
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d7kpya_ - Chain 'B':
Compound: histone acetyltransferase
Species: Homo sapiens [TaxId:9606]
Gene: Crebbp
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d7kpyb_ - Heterogens: WU1, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>7kpyA (A:)
kkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrk
ldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>7kpyA (A:)
kifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkl
dtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
- Chain 'B':
Sequence, based on SEQRES records: (download)
>7kpyB (B:)
kkifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrk
ldtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg
Sequence, based on observed residues (ATOM records): (download)
>7kpyB (B:)
kifkpeelrqalmptlealyrqdpeslpfrqpvdpqllgipdyfdivknpmdlstikrkl
dtgqyqepwqyvddvwlmfnnawlynrktsrvykfcsklaevfeqeidpvmqslg