PDB entry 7ki8
View 7ki8 on RCSB PDB site
Description: Crystal Structure of Dihydrofolate reductase (DHFR) from Mycobacterium ulcerans Agy99 in complex with NADP and inhibitor SDDC-0001580
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: SSGCID, SDDC, inhibitor, Structural Genomics, Seattle Structural Genomics Center for Infectious Disease, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2020-10-23, released
2021-07-07
The last revision prior to the SCOPe 2.08 freeze date was dated
2021-07-07, with a file datestamp of
2021-07-02.
Experiment type: XRAY
Resolution: 1.25 Å
R-factor: N/A
AEROSPACI score: 0.7
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: dihydrofolate reductase
Species: Mycobacterium ulcerans (strain Agy99) [TaxId:362242]
Gene: dfrA, MUL_2179
Database cross-references and differences (RAF-indexed):
- Uniprot A0PQG8 (8-172)
- expression tag (0-7)
- engineered mutation (96)
- engineered mutation (103)
Domains in SCOPe 2.08: d7ki8a_ - Heterogens: WFA, NAP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>7ki8A (A:)
mahhhhhhmtsvgliwaqstsgvigrdggipwrlpedlahfkrltmghtvvmgrrtwdsl
paahrplpgrrnvvvtrqtglvahgaqvvgsleqalspaepdaatwviggaqiyalalpl
anrcevtevdvdlppededalapvldqtwagtsgewlvsrsglryrmhsyrrl
Sequence, based on observed residues (ATOM records): (download)
>7ki8A (A:)
svgliwaqstsgvigrdggipwrlpedlahfkrltmghtvvmgrrtwdslpaahrplpgr
rnvvvtrqtglvahgaqvvgsleqalspaepdaatwviggaqiyalalplanrcevtevd
vdlppededalapvldqtwagtsgewlvsrsglryrmhsyrrl