PDB entry 7dua
View 7dua on RCSB PDB site
Description: Crystal structure of human Proto-oncogene tyrosine-protein kinase receptor Ret in complex with 4-amino-7-(1-methylcyclopropyl)-N-(5-methyl-1H-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide
Class: transferase
Keywords: tyrosine-protein kinase, transferase
Deposited on
2021-01-08, released
2022-01-12
The last revision prior to the SCOPe 2.08 freeze date was dated
2022-01-12, with a file datestamp of
2022-01-07.
Experiment type: XRAY
Resolution: 1.64 Å
R-factor: N/A
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: proto-oncogene tyrosine-protein kinase receptor ret
Species: Homo sapiens [TaxId:9606]
Gene: RET, CDHF12, CDHR16, PTC, RET51
Database cross-references and differences (RAF-indexed):
- Chain 'B':
Compound: proto-oncogene tyrosine-protein kinase receptor ret
Species: Homo sapiens [TaxId:9606]
Gene: RET, CDHF12, CDHR16, PTC, RET51
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d7duab1, d7duab2 - Heterogens: HJ0, HOH
PDB Chain Sequences:
- Chain 'A':
No sequence available.
- Chain 'B':
Sequence, based on SEQRES records: (download)
>7duaB (B:)
gplslsvdafkiledpkwefprknlvlgktlgegefgkvvkatafhlkgragyttvavkm
lkenaspselrdllsefnvlkqvnhphviklygacsqdgpllliveyakygslrgflres
rkvgpgylgsggsrnsssldhpderaltmgdlisfawqisqgmqylaemklvhrdlaarn
ilvaegrkmkisdfglsrdvyeedsyvkrsqgripvkwmaieslfdhiyttqsdvwsfgv
llweivtlggnpypgipperlfnllktghrmerpdncseemyrlmlqcwkqepdkrpvfa
diskdlekmmvkrr
Sequence, based on observed residues (ATOM records): (download)
>7duaB (B:)
gplslsvdafkipkwefprknlvlgktlgegefgkvvkatafhlkgragyttvavkmlke
naspselrdllsefnvlkqvnhphviklygacsqdgpllliveyakygslrgflresltm
gdlisfawqisqgmqylaemklvhrdlaarnilvaegrkmkisdfglsrdvqgripvkwm
aieslfdhiyttqsdvwsfgvllweivtlggnpypgipperlfnllktghrmerpdncse
emyrlmlqcwkqepdkrpvfadiskdlekmmvkr