PDB entry 7aw4

View 7aw4 on RCSB PDB site
Description: mertk kinase domain with type 3 inhibitor from a dna-encoded library
Deposited on 2020-11-06, released 2021-03-03
The last revision was dated 2021-04-07, with a file datestamp of 2021-04-02.
Experiment type: XRAY
Resolution: 1.98 Å
R-factor: N/A
AEROSPACI score: 0.4 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Tyrosine-protein kinase Mer
    Species: Homo sapiens [TaxId:9606]
    Gene: MERTK, MER
    Database cross-references and differences (RAF-indexed):
  • Chain 'B':
    Compound: Tyrosine-protein kinase Mer
    Species: Homo sapiens [TaxId:9606]
    Gene: MERTK, MER
    Database cross-references and differences (RAF-indexed):
  • Heterogens: S5E, CL, EDO, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >7aw4A (A:)
    mgsshhhhhhssglvprgseelqnkledvvidrnllilgkilgegefgsvmegnlkqedg
    tslkvavktmkldnssqreieeflseaacmkdfshpnvirllgvciemssqgipkpmvil
    pfmkygdlhtyllysrletgpkhiplqtllkfmvdialgmeylsnrnflhrdlaarncml
    rddmtvcvadfglskkiysgdyyrqgriakmpvkwiaiesladrvytsksdvwafgvtmw
    eiatrgmtpypgvqnhemydyllhghrlkqpedcldelyeimyscwrtdpldrptfsvlr
    lqleklleslpdv
    

    Sequence, based on observed residues (ATOM records):
    >7aw4A (A:)
    kledvvidrnllilgkilgegefgsvmegnlkqedgtslkvavktmkldnssqreieefl
    seaacmkdfshpnvirllgvciepkpmvilpfmkygdlhtyllysrletgpkhiplqtll
    kfmvdialgmeylsnrnflhrdlaarncmlrddmtvcvadfglspvkwiaiesladrvyt
    sksdvwafgvtmweiatrgmtpypgvqnhemydyllhghrlkqpedcldelyeimyscwr
    tdpldrptfsvlrlqleklleslp
    

  • Chain 'B':
    Sequence, based on SEQRES records:
    >7aw4B (B:)
    mgsshhhhhhssglvprgseelqnkledvvidrnllilgkilgegefgsvmegnlkqedg
    tslkvavktmkldnssqreieeflseaacmkdfshpnvirllgvciemssqgipkpmvil
    pfmkygdlhtyllysrletgpkhiplqtllkfmvdialgmeylsnrnflhrdlaarncml
    rddmtvcvadfglskkiysgdyyrqgriakmpvkwiaiesladrvytsksdvwafgvtmw
    eiatrgmtpypgvqnhemydyllhghrlkqpedcldelyeimyscwrtdpldrptfsvlr
    lqleklleslpdv
    

    Sequence, based on observed residues (ATOM records):
    >7aw4B (B:)
    qnkledvvidrnllilgkilgegefgsvmegnlkqedgtslkvavktmkeieeflseaac
    mkdfshpnvirllgvciekpmvilpfmkygdlhtyllysrletgpkhiplqtllkfmvdi
    algmeylsnrnflhrdlaarncmlrddmtvcvadfglpvkwiaiesladrvytsksdvwa
    fgvtmweiatrgmtpypgvqnhemydyllhghrlkqpedcldelyeimyscwrtdpldrp
    tfsvlrlqleklleslp