PDB entry 7ah5

View 7ah5 on RCSB PDB site
Description: Crystal structure of indoleamine 2,3-dioxygenase 1 (IDO1) in complex with ferric heme and MMG-0706
Class: oxidoreductase
Keywords: Oxidoreductase, Dioxygenase, Heme-containing enzyme, Structure-based drug design, IDO1 inhibitor, Triazole, Small-molecule inhibitor
Deposited on 2020-09-24, released 2021-02-17
The last revision prior to the SCOPe 2.07 freeze date was dated 2021-03-10, with a file datestamp of 2021-03-05.
Experiment type: XRAY
Resolution: 2.9 Å
R-factor: N/A
AEROSPACI score: 0.22 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Indoleamine 2,3-dioxygenase 1
    Species: Homo sapiens [TaxId:9606]
    Gene: IDO1, IDO, INDO
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d7ah5a_
  • Chain 'B':
    Compound: Indoleamine 2,3-dioxygenase 1
    Species: Homo sapiens [TaxId:9606]
    Gene: IDO1, IDO, INDO
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d7ah5b_
  • Heterogens: RCQ, HEM

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >7ah5A (A:)
    mgsshhhhhhssglvprgshmasamenswtiskeyhideevgfalpnpqenlpdfyndwm
    fiakhlpdliesgqlrerveklnmlsidhltdhksqrlarlvlgcitmayvwgkghgdvr
    kvlprniavpycqlskklelppilvyadcvlanwkkkdpnkpltyenmdvlfsfrdgdcs
    kgfflvsllveiaaasaikviptvfkamqmqerdtllkalleiasclekalqvfhqihdh
    vnpkaffsvlriylsgwkgnpqlsdglvyegfwedpkefaggsagqssvfqcfdvllgiq
    qtaggghaaqflqdmrrymppahrnflcslesnpsvrefvlskgdaglreaydacvkalv
    slrsyhlqivtkyilipasqqpkenktsedpskleakgtggtdlmnflktvrstteksll
    keg
    

    Sequence, based on observed residues (ATOM records): (download)
    >7ah5A (A:)
    keyhideevgfalpnpqenlpdfyndwmfiakhlpdliesgqlrerveklnmlsidhltd
    hksqrlarlvlgcitmayvwgkghgdvrkvlprniavpycqlskklelppilvyadcvla
    nwkkkdpnkpltyenmdvlfsfrdgdcskgfflvsllveiaaasaikviptvfkamqmqe
    rdtllkalleiasclekalqvfhqihdhvnpkaffsvlriylsgwkgnpqlsdglvyegf
    wedpkefaggsagqssvfqcfdvllgiqqtaggghaaqflqdmrrymppahrnflcsles
    npsvrefvlskgdaglreaydacvkalvslrsyhlqivtkyilipasqqgtdlmnflktv
    rstteksllke
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >7ah5B (B:)
    mgsshhhhhhssglvprgshmasamenswtiskeyhideevgfalpnpqenlpdfyndwm
    fiakhlpdliesgqlrerveklnmlsidhltdhksqrlarlvlgcitmayvwgkghgdvr
    kvlprniavpycqlskklelppilvyadcvlanwkkkdpnkpltyenmdvlfsfrdgdcs
    kgfflvsllveiaaasaikviptvfkamqmqerdtllkalleiasclekalqvfhqihdh
    vnpkaffsvlriylsgwkgnpqlsdglvyegfwedpkefaggsagqssvfqcfdvllgiq
    qtaggghaaqflqdmrrymppahrnflcslesnpsvrefvlskgdaglreaydacvkalv
    slrsyhlqivtkyilipasqqpkenktsedpskleakgtggtdlmnflktvrstteksll
    keg
    

    Sequence, based on observed residues (ATOM records): (download)
    >7ah5B (B:)
    skeyhideevgfalpnpqenlpdfyndwmfiakhlpdliesgqlrerveklnmlsidhlt
    dhksqrlarlvlgcitmayvwgkghgdvrkvlprniavpycqlskklelppilvyadcvl
    anwkkkdpnkpltyenmdvlfsfrdgdcskgfflvsllveiaaasaikviptvfkamqmq
    erdtllkalleiasclekalqvfhqihdhvnpkaffsvlriylsgwkgnpqlsdglvyeg
    fwedpkefaggsagqssvfqcfdvllgiqqtaggghaaqflqdmrrymppahrnflcsle
    snpsvrefvlskgdaglreaydacvkalvslrsyhlqivtkyilipasqggtdlmnflkt
    vrstteksllk