PDB entry 7aaz

View 7aaz on RCSB PDB site
Description: crystal structure of mertk in complex with a type 1.5 aminopyridine inhibitor
Deposited on 2020-09-05, released 2020-11-04
The last revision was dated 2020-12-09, with a file datestamp of 2020-12-04.
Experiment type: XRAY
Resolution: 1.86 Å
R-factor: N/A
AEROSPACI score: 0.44 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Tyrosine-protein kinase Mer
    Species: Homo sapiens [TaxId:9606]
    Gene: MERTK, MER
    Database cross-references and differences (RAF-indexed):
  • Heterogens: R6K, CL, EDO, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >7aazA (A:)
    gseelqnkledvvidrnllilgkilgegefgsvmegnlkqedgtslkvavktmkldnssq
    reieeflseaacmkdfshpnvirllgvciemssqgipkpmvilpfmkygdlhtyllysrl
    etgpkhiplqtllkfmvdialgmeylsnrnflhrdlaarncmlrddmtvcvadfglskki
    ysgdyyrqgriakmpvkwiaiesladrvytsksdvwafgvtmweiatrgmtpypgvqnhe
    mydyllhghrlkqpedcldelyeimyscwrtdpldrptfsvlrlqleklleslpdv
    

    Sequence, based on observed residues (ATOM records):
    >7aazA (A:)
    qnkledvvidrnllilgkilgegefgsvmegnlkqedgtslkvavktmkldnssqreiee
    flseaacmkdfshpnvirllgvciemssqgipkpmvilpfmkygdlhtyllysrletgpk
    hiplqtllkfmvdialgmeylsnrnflhrdlaarncmlrddmtvcvadfglskkiysgdy
    yrqgriakmpvkwiaiesladrvytsksdvwafgvtmweiatrgmtpypgvqnhemydyl
    lhghrlkqpedcldelyeimyscwrtdpldrptfsvlrlqleklleslpd