PDB entry 6v6l
View 6v6l on RCSB PDB site
Description: Co-structure of human glycogen synthase kinase beta with 1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-one
Class: transferase
Keywords: kinase, TRANSFERASE
Deposited on
2019-12-05, released
2020-01-15
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-02-05, with a file datestamp of
2020-01-31.
Experiment type: XRAY
Resolution: 2.19 Å
R-factor: N/A
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Glycogen synthase kinase-3 beta
Species: Homo sapiens [TaxId:9606]
Gene: GSK3B
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6v6la_ - Heterogens: QQA, PO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6v6lA (A:)
msgrprttsfaesckpvqqpsafgsmkvsrdkdgskvttvvatpgqgpdrpqevsytdtk
vigngsfgvvyqaklcdsgelvaikkvlqdkrfknrelqimrkldhcnivrlryffyssg
ekkdevylnlvldyvpetvyrvarhysrakqtlpviyvklymyqlfrslayihsfgichr
dikpqnllldpdtavlklcdfgsakqlvrgepnvsyicsryyrapelifgatdytssidv
wsagcvlaelllgqpifpgdsgvdqlveiikvlgtptreqiremnpnytefkfpqikahp
wtkvfrprtppeaialcsrlleytptarltpleacahsffdelrdpnvklpngrdtpalf
nfttqelssnpplatilipphariqaaastptnataasdantgdrgqtnnaasasasnst
Sequence, based on observed residues (ATOM records): (download)
>6v6lA (A:)
vttvvatpgqgpdrpqevsytdtkvigngsfgvvyqaklcdsgelvaikkvlqdkrelqi
mrkldhcnivrlryffyssgekkdevylnlvldyvpetvyrvarhysrakqtlpviyvkl
ymyqlfrslayihsfgichrdikpqnllldpdtavlklcdfgsakqlvrgepnvsyicsr
yyrapelifgatdytssidvwsagcvlaelllgqpifpgdsgvdqlveiikvlgtptreq
iremnpnytefkfpqikahpwtkvfrprtppeaialcsrlleytptarltpleacahsff
delrdpnvklpngrdtpalfnfttqelssnpplatilipphari