PDB entry 6tcu

View 6tcu on RCSB PDB site
Description: Glycogen synthase kinase-3 beta (GSK3b) in complex with ligand 1
Class: transferase
Keywords: gsk3beta kinase, transferase, inhibitor, proteros
Deposited on 2019-11-06, released 2020-09-16
The last revision prior to the SCOPe 2.08 freeze date was dated 2020-09-16, with a file datestamp of 2020-09-11.
Experiment type: XRAY
Resolution: 2.14 Å
R-factor: N/A
AEROSPACI score: 0.37 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glycogen synthase kinase-3 beta
    Species: Homo sapiens [TaxId:9606]
    Gene: GSK3B
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6tcua_
  • Heterogens: N1Q, ACT, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6tcuA (A:)
    gamskvttvvatpgqgpdrpqevsytdtkvigngsfgvvyqaklcdsgelvaikkvlqdk
    rfknrelqimrkldhcnivrlryffyssgekkdevylnlvldyvpetvyrvarhysrakq
    tlpviyvklymyqlfrslayihsfgichrdikpqnllldpdtavlklcdfgsakqlvrge
    pnvsyicsryyrapelifgatdytssidvwsagcvlaelllgqpifpgdsgvdqlveiik
    vlgtptreqiremnpnytefkfpqikahpwtkvfrprtppeaialcsrlleytptarltp
    leacahsffdelrdpnvklpngrdtpalfnfttqelssnpplatilipphariqa
    

    Sequence, based on observed residues (ATOM records): (download)
    >6tcuA (A:)
    skvttvvatpgqgpdrpqevsytdtkvigngsfgvvyqaklcdsgelvaikkvlqdkrfk
    nrelqimrkldhcnivrlryffyssgekkdevylnlvldyvpetvyrvarhysrakqtlp
    viyvklymyqlfrslayihsfgichrdikpqnllldpdtavlklcdfgsakqlvrgepnv
    syicsryyrapelifgatdytssidvwsagcvlaelllgqpifpgdsgvdqlveiikvlg
    tptreqiremnpnytefkfpqikahpwtkvfrprtppeaialcsrlleytptarltplea
    cahsffdelrdpnvklpngrdtpalfnfttqelssnpplatilipphari