PDB entry 6t6f

View 6t6f on RCSB PDB site
Description: Crystal structure of human calmodulin-dependent protein kinase 1D (CAMK1D) bound to compound 8 (CS275)
Class: transferase
Keywords: Inhibitor, Complex, Kinase, Structural Genomics, Structural Genomics Consortium, SGC, TRANSFERASE
Deposited on 2019-10-18, released 2020-01-15
The last revision prior to the SCOPe 2.08 freeze date was dated 2020-01-15, with a file datestamp of 2020-01-10.
Experiment type: XRAY
Resolution: 1.97 Å
R-factor: N/A
AEROSPACI score: 0.32 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: calcium/calmodulin-dependent protein kinase type 1d
    Species: Homo sapiens [TaxId:9606]
    Gene: CAMK1D, CAMKID
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6t6fa_
  • Chain 'B':
    Compound: calcium/calmodulin-dependent protein kinase type 1d
    Species: Homo sapiens [TaxId:9606]
    Gene: CAMK1D, CAMKID
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6t6fb_
  • Heterogens: MMW, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6t6fA (A:)
    smsswkkqaedikkifefketlgtgafsevvlaeekatgklfavkcipkkalkgkessie
    neiavlrkikhenivalediyespnhlylvmqlvsggelfdrivekgfytekdastlirq
    vldavyylhrmgivhrdlkpenllyysqdeeskimisdfglskmegkgdvmstacgtpgy
    vapevlaqkpyskavdcwsigviayillcgyppfydendsklfeqilkaeyefdspywdd
    isdsakdfirnlmekdpnkrytceqaarhpwiagdtalnknihesvsaqirknfakskwr
    qafnatavvrhmrklhlgssld
    

    Sequence, based on observed residues (ATOM records): (download)
    >6t6fA (A:)
    wkkqaedikkifefketlgtgafsevvlaeekatgklfavkcipkkalkgkessieneia
    vlrkikhenivalediyespnhlylvmqlvsggelfdrivekgfytekdastlirqvlda
    vyylhrmgivhrdlkpenllyysqdeeskimisdfglspgyvapevlaqkpyskavdcws
    igviayillcgyppfydendsklfeqilkaeyefdspywddisdsakdfirnlmekdpnk
    rytceqaarhpwiagdtalnknihesvsaqirknfakhmrklhlgssld
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >6t6fB (B:)
    smsswkkqaedikkifefketlgtgafsevvlaeekatgklfavkcipkkalkgkessie
    neiavlrkikhenivalediyespnhlylvmqlvsggelfdrivekgfytekdastlirq
    vldavyylhrmgivhrdlkpenllyysqdeeskimisdfglskmegkgdvmstacgtpgy
    vapevlaqkpyskavdcwsigviayillcgyppfydendsklfeqilkaeyefdspywdd
    isdsakdfirnlmekdpnkrytceqaarhpwiagdtalnknihesvsaqirknfakskwr
    qafnatavvrhmrklhlgssld
    

    Sequence, based on observed residues (ATOM records): (download)
    >6t6fB (B:)
    wkkqaedikkifefketlgtgafsevvlaeekatgklfavkcipkkalkgkessieneia
    vlrkikhenivalediyespnhlylvmqlvsggelfdrivekgfytekdastlirqvlda
    vyylhrmgivhrdlkpenllyysqdeeskimisdfgpgyvapevlaqkpyskavdcwsig
    viayillcgyppfydendsklfeqilkaeyefdspywddisdsakdfirnlmekdpnkry
    tceqaarhpwiagdtalnknihesvsaqirknfakmrklhlgssld