PDB entry 6sp9
View 6sp9 on RCSB PDB site
Description: Fragment KCL802 in complex with MAP kinase p38-alpha
Class: transferase
Keywords: FBDD, Fragment Based Drug Design, P38, MAPK14, Kinase, Transferase., TRANSFERASE
Deposited on
2019-08-31, released
2019-10-02
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-10-14, with a file datestamp of
2020-10-09.
Experiment type: XRAY
Resolution: 1.22 Å
R-factor: N/A
AEROSPACI score: 0.72
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Mus musculus [TaxId:10090]
Gene: Mapk14, Crk1, Csbp1, Csbp2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6sp9a_ - Heterogens: LOT, SB4, CA, DMS, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6sp9A (A:)
gmsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktghrvavkklsrpf
qsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkc
qkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglarhtddem
tgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlv
gtpgaellkkissesarnyiqslaqmpkmnfanvfiganplavdllekmlvldsdkrita
aqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeeme
s
Sequence, based on observed residues (ATOM records): (download)
>6sp9A (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktghrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltd
dhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfgarhtyvatrwyrap
eimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkis
sesarnyiqslaqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqy
hdpddepvadpydqsfesrdllidewksltydevisfvpppldqeeme