PDB entry 6sd9

View 6sd9 on RCSB PDB site
Description: Crystal structure of wild-type cMET bound by foretinib
Class: transferase
Keywords: Kinase, inhibitor, transferase
Deposited on 2019-07-26, released 2019-08-14
The last revision prior to the SCOPe 2.08 freeze date was dated 2019-10-02, with a file datestamp of 2019-09-27.
Experiment type: XRAY
Resolution: 2.35 Å
R-factor: N/A
AEROSPACI score: 0.23 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Hepatocyte growth factor receptor
    Species: Homo sapiens [TaxId:9606]
    Gene: MET
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6sd9a_
  • Heterogens: 88Z, CL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6sd9A (A:)
    gdsdisspllqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtl
    ldndgkkihcavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvl
    pymkhgdlrnfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekft
    vkvadfglardmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelm
    trgappypdvntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsri
    saifstfig
    

    Sequence, based on observed residues (ATOM records): (download)
    >6sd9A (A:)
    lvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihcavkslnrevsqflt
    egiimkdfshpnvlsllgiclplvvlpymkhgdlrnfirnethnptvkdligfglqvakg
    mkylaskkfvhrdlaarncmldekftvkvadfglareyystgaklpvkwmaleslqtqkf
    ttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdplyevmlkcw
    hpkaemrpsfselvsrisaifstfi