PDB entry 6sbt

View 6sbt on RCSB PDB site
Description: Structure of GluK1 ligand-binding domain (S1S2) in complex with N-(7-(1H-imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl benzamide at 2.3 A resolution
Class: membrane protein
Keywords: kainate receptor ligand-binding domain, GluK1-S1S2, antagonist, membrane protein
Deposited on 2019-07-22, released 2019-10-30
The last revision prior to the SCOPe 2.08 freeze date was dated 2019-11-27, with a file datestamp of 2019-11-22.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: N/A
AEROSPACI score: 0.25 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glutamate receptor ionotropic, kainate 1
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Grik1, Glur5
    Database cross-references and differences (RAF-indexed):
    • Uniprot P22756 (Start-115)
      • variant (33)
      • linker (116-117)
    • Uniprot P22756 (118-End)
    Domains in SCOPe 2.08: d6sbta_
  • Heterogens: L5H, SO4, CL, GOL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6sbtA (A:)
    ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
    ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
    dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
    lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
    gklhmmkekwwrgngcp
    

    Sequence, based on observed residues (ATOM records): (download)
    >6sbtA (A:)
    rtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyga
    qndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsa
    ddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvltt
    dyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegkl
    hmmkekwwr