PDB entry 6s9w

View 6s9w on RCSB PDB site
Description: crystal structure of akt1 in complex with covalent-allosteric akt inhibitor 16a
Deposited on 2019-07-15, released 2019-10-16
The last revision was dated 2019-12-25, with a file datestamp of 2019-12-20.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: N/A
AEROSPACI score: 0.25 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: RAC-alpha serine/threonine-protein kinase
    Species: Homo sapiens [TaxId:9606]
    Gene: AKT1, PKB, RAC
    Database cross-references and differences (RAF-indexed):
  • Heterogens: L1Z, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >6s9wA (A:)
    gsdvaivkegwlhkrgeyiktwrpryfllkndgtfigykerpqdvdqreaplnnfsvaqc
    qlmkterprpntfiirclqwttviertfhvetpeereewttaiqtvadglkkqaaaemdf
    rsgspsdnsgaeemevslakpkhrvtmnefeylkllgkgtfgkvilvkekatgryyamki
    lkkevivakdevahtltenrvlqnsrhpfltalkysfqthdrlcfvmeyanggelffhls
    rervfsedrarfygaeivsaldylhseknvvyrdlklenlmldkdghikitdfglckegi
    kdgatmktfcgtpeylapevledndygravdwwglgvvmyemmcgrlpfynqdheklfel
    ilmeeirfprtlgpeaksllsgllkkdpkqrlgggsedakeimqhrffagivwqhvyekk
    lsppfkpqvtsetdtryfdeeftaqm
    

    Sequence, based on observed residues (ATOM records):
    >6s9wA (A:)
    dvaivkegwlhkrgeyiktwrpryfllkndgtfigykerpqdvdqreaplnnfsvaqcql
    mkterprpntfiirclqwttviertfhvetpeereewttaiqtvadglkkkhrvtmnefe
    ylkllgkgtfgkvilvkekatgryyamkilkkevivakdevahtltenrvlqnsrhpflt
    alkysfqthdrlcfvmeyanggelffhlsrervfsedrarfygaeivsaldylhseknvv
    yrdlklenlmldkdghikitdfglckegikatmktfcgtpeylapevledndygravdww
    glgvvmyemmcgrlpfynqdheklfelilmeeirfprtlgpeaksllsgllkkdpkqrlg
    ggsedakeimqhrffagivwqhvyekklsppfkpqvtsetdtryfdeefta