PDB entry 6pg9

View 6pg9 on RCSB PDB site
Description: WDR5delta23 bound to N-(4-(5-(hydroxymethyl)-1H-imidazol-2-yl)butyl)benzamide
Class: PROTEIN BINDING/Inhibitor
Keywords: Inhibitor, Scaffolding Protein, B-propellor, Chromatin regulator, PROTEIN BINDING, PROTEIN BINDING-Inhibitor complex
Deposited on 2019-06-24, released 2019-12-11
The last revision prior to the SCOPe 2.08 freeze date was dated 2019-12-11, with a file datestamp of 2019-12-06.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: N/A
AEROSPACI score: 0.38 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: WD repeat-containing protein 5
    Species: Homo sapiens [TaxId:9606]
    Gene: WDR5, BIG3
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6pg9a_
  • Chain 'B':
    Compound: WD repeat-containing protein 5
    Species: Homo sapiens [TaxId:9606]
    Gene: WDR5, BIG3
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d6pg9b_
  • Heterogens: OH1, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6pg9A (A:)
    gsatqskptpvkpnyalkftlaghtkavssvkfspngewlasssadklikiwgaydgkfe
    ktisghklgisdvawssdsnllvsasddktlkiwdvssgkclktlkghsnyvfccnfnpq
    snlivsgsfdesvriwdvktgkclktlpahsdpvsavhfnrdgslivsssydglcriwdt
    asgqclktlidddnppvsfvkfspngkyilaatldntlklwdyskgkclktytghkneky
    cifanfsvtggkwivsgsednlvyiwnlqtkeivqklqghtdvvistachpteniiasaa
    lendktiklwksdc
    

    Sequence, based on observed residues (ATOM records): (download)
    >6pg9A (A:)
    vkpnyalkftlaghtkavssvkfspngewlasssadklikiwgaydgkfektisghklgi
    sdvawssdsnllvsasddktlkiwdvssgkclktlkghsnyvfccnfnpqsnlivsgsfd
    esvriwdvktgkclktlpahsdpvsavhfnrdgslivsssydglcriwdtasgqclktli
    dddnppvsfvkfspngkyilaatldntlklwdyskgkclktytghknekycifanfsvtg
    gkwivsgsednlvyiwnlqtkeivqklqghtdvvistachpteniiasaalendktiklw
    ksdc
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >6pg9B (B:)
    gsatqskptpvkpnyalkftlaghtkavssvkfspngewlasssadklikiwgaydgkfe
    ktisghklgisdvawssdsnllvsasddktlkiwdvssgkclktlkghsnyvfccnfnpq
    snlivsgsfdesvriwdvktgkclktlpahsdpvsavhfnrdgslivsssydglcriwdt
    asgqclktlidddnppvsfvkfspngkyilaatldntlklwdyskgkclktytghkneky
    cifanfsvtggkwivsgsednlvyiwnlqtkeivqklqghtdvvistachpteniiasaa
    lendktiklwksdc
    

    Sequence, based on observed residues (ATOM records): (download)
    >6pg9B (B:)
    vkpnyalkftlaghtkavssvkfspngewlasssadklikiwgaydgkfektisghklgi
    sdvawssdsnllvsasddktlkiwdvssgkclktlkghsnyvfccnfnpqsnlivsgsfd
    esvriwdvktgkclktlpahsdpvsavhfnrdgslivsssydglcriwdtasgqclktli
    dddnppvsfvkfspngkyilaatldntlklwdyskgkclktytghknekycifanfsvtg
    gkwivsgsednlvyiwnlqtkeivqklqghtdvvistachpteniiasaalendktiklw
    ksdc