PDB entry 6pda
View 6pda on RCSB PDB site
Description: Crystal structure of MYST acetyltransferase domain in complex with inhibitor 74
Class: transferase/transferase inhibitor
Keywords: Inhibitor, Complex, MYST, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2019-06-18, released
2020-04-01
The last revision prior to the SCOPe 2.07 freeze date was dated
2020-04-01, with a file datestamp of
2020-03-27.
Experiment type: XRAY
Resolution: 2.45 Å
R-factor: N/A
AEROSPACI score: 0.22
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Histone acetyltransferase KAT8
Species: Homo sapiens [TaxId:9606]
Gene: KAT8, MOF, MYST1, PP7073
Database cross-references and differences (RAF-indexed):
- Uniprot Q9H7Z6 (0-271)
- conflict (72)
- engineered mutation (138)
- engineered mutation (141-142)
- engineered mutation (153)
- engineered mutation (190)
- conflict (195)
Domains in SCOPe 2.07: d6pdaa_ - Heterogens: O9J, ZN, NA, GOL, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6pdaA (A:)
kyvdkihignyeidawyfspfpedygkqpklwlceyclkymkyeksyrfhlgqcqwrqpp
gkeiyrksnisvhevdgkdhkiycqnlcllaklfldhktlyfdvepfvfyiltevdrqga
hivgyfskekespdgnnvscimilppyqrrgygrfliafsyelsklestvgspekplsdl
gklsyrsywssvllenlrdfrgtlsikdlsqmtsitqndiistlqslnmvkywkgqhvic
vtpklveehlksaqykkppitvdsvclkwapp
Sequence, based on observed residues (ATOM records): (download)
>6pdaA (A:)
kyvdkihignyeidawyfspfpedygkqpklwlceyclkymkyeksyrfhlgqcqwrqpp
gkeiyrksnisvhevdgkdhkiycqnlcllaklfldhktlyfdvepfvfyiltevdrqga
hivgyfskekespdgnnvscimilppyqrrgygrfliafsyelsklestvgspekplsdl
gklsyrsywssvllenlrdlsikdlsqmtsitqndiistlqslnmvkywkgqhvicvtpk
lveehlksaqykkppitvdsvclkwapp