PDB entry 6owi
View 6owi on RCSB PDB site
Description: Crystal structure of MYST acetyltransferase domain in complex with inhibitor 85
Class: transferase/transerase inhibitor
Keywords: Inhibitor, Complex, MYST, TRANSFERASE, TRANSFERASE-TRANSERASE INHIBITOR complex
Deposited on
2019-05-09, released
2020-04-01
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-05-27, with a file datestamp of
2020-05-22.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: N/A
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Histone acetyltransferase KAT8
Species: Homo sapiens [TaxId:9606]
Gene: KAT8, MOF, MYST1, PP7073
Database cross-references and differences (RAF-indexed):
- Uniprot Q9H7Z6
- conflict (73)
- engineered mutation (139)
- engineered mutation (142-143)
- engineered mutation (154)
- conflict (196)
Domains in SCOPe 2.08: d6owia_ - Heterogens: NB7, ZN, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6owiA (A:)
vkyvdkihignyeidawyfspfpedygkqpklwlceyclkymkyeksyrfhlgqcqwrqp
pgkeiyrksnisvhevdgkdhkiycqnlcllaklfldhktlyfdvepfvfyiltevdrqg
ahivgyfskekespdgnnvscimilppyqrrgygrfliafsyelsklestvgspekplsd
lgklsyrsywswvllenlrdfrgtlsikdlsqmtsitqndiistlqslnmvkywkgqhvi
cvtpklveehlksaqykkppitvdsvclkwapp
Sequence, based on observed residues (ATOM records): (download)
>6owiA (A:)
kyvdkihignyeidawyfspfpedygkqpklwlceyclkymkyeksyrfhlgqcqwrqpp
gkeiyrksnisvhevdgkdhkiycqnlcllaklfldhktlyfdvepfvfyiltevdrqga
hivgyfskekespdgnnvscimilppyqrrgygrfliafsyelsklestvgspekplsdl
gklsyrsywswvllenlrdftlsikdlsqmtsitqndiistlqslnmvkywkgqhvicvt
pklveehlksaqykkppitvdsvclkwap