PDB entry 6o9o

View 6o9o on RCSB PDB site
Description: crystal structure of smyd3 with potent and selective isoxazole amide inhibitor 1
Deposited on 2019-03-14, released 2020-03-18
The last revision was dated 2020-03-18, with a file datestamp of 2020-03-13.
Experiment type: XRAY
Resolution: 1.59 Å
R-factor: N/A
AEROSPACI score: 0.45 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Histone-lysine N-methyltransferase SMYD3
    Species: Homo sapiens [TaxId:9606]
    Gene: SMYD3, ZMYND1, ZNFN3A1
    Database cross-references and differences (RAF-indexed):
    • Uniprot Q9H7B4 (Start-431)
      • conflict (16)
  • Heterogens: ZN, MG, GOL, SAH, LUP, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >6o9oA (A:)
    gsftmeplkvekfatanrgnglravtplrpgellfrsdplaytvckgsrgvvcdrcllgk
    eklmrcsqcrvakycsakcqkkawpdhkreckclksckpryppdsvrllgrvvfklmdga
    pseseklysfydlesninkltedkkeglrqlvmtfqhfmreeiqdasqlppafdlfeafa
    kvicnsfticnaemqevgvglypsisllnhscdpncsivfngphlllravrdievgeelt
    icyldmlmtseerrkqlrdqycfecdcfrcqtqdkdadmltgdeqvwkevqeslkkieel
    kahwkweqvlamcqaiissnserlpdiniyqlkvldcamdacinlglleealfygtrtme
    pyriffpgshpvrgvqvmkvgklqlhqgmfpqamknlrlafdimrvthgrehsliedlil
    lleecdaniras
    

    Sequence, based on observed residues (ATOM records):
    >6o9oA (A:)
    plkvekfatanrgnglravtplrpgellfrsdplaytvckgsrgvvcdrcllgkeklmrc
    sqcrvakycsakcqkkawpdhkreckclksckpryppdsvrllgrvvfklmdgapsesek
    lysfydlesninkltedkkeglrqlvmtfqhfmreeiqdasqlppafdlfeafakvicns
    fticnaemqevgvglypsisllnhscdpncsivfngphlllravrdievgeelticyldm
    lmtseerrkqlrdqycfecdcfrcqtqdkdadmltgdeqvwkevqeslkkieelkahwkw
    eqvlamcqaiissnserlpdiniyqlkvldcamdacinlglleealfygtrtmepyriff
    pgshpvrgvqvmkvgklqlhqgmfpqamknlrlafdimrvthgrehsliedlillleecd
    aniras